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       5-HT(5-Hydroxytryptamine,5-羥色胺)神經遞質主要分布于松果體和下丘腦,可參與食欲、體溫調節,情緒,心血管功能,內分泌和抑郁等生理功能的調節。5-HT通過激動不同的5-HT受體,可具有不同藥理作用,因此,5-HT受體拮抗劑成為藥物設計的研究熱點[1][2]。百靈威作為專業試劑供應商,提供多種5-HT受體拮抗劑,為您的科研助力加油!

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    產品編號

    中英文名稱

    CAS

    規格

    384285

    Granisetron hydrochloride, 98%, a serotonin 5-HT3 receptor antagonist

    鹽酸格拉司瓊, 98%, 5-HT3受體拮抗劑

    107007-99-8

    200 mg

    1 g

    283801

    Ketanserin, 99%, a specific 5-HT2A serotonin receptor antagonist

    凱他色林, 99%, 特異性的5-HT2A 5-羥色胺受體拮抗劑

    74050-98-9

    250 mg

    1 g

    185928

    Lamotrigine, 98%, Novel anticonvulsant drug for inhibition of 5-HT

    拉莫三嗪, 98%, 抑制5-羥色胺(5-HT)吸收

    84057-84-1

    1 g

    5 g

    574335

    Mirtazapine, 99%, 5-HT Receptor

    米爾塔扎平, 99%, 5-HT受體抑制劑

    85650-52-8

    100 mg

    496697

    Olanzapine, 99%, High affinity for 5-HT2 serotonin and D2 dopamine receptor antagonist

    奧氮平, 99%, 5-HT2D2受體高親和性拮抗劑

    132539-06-1

    1 g

    5 g

    977215

    Paliperidone, 99%, potent D2 and 5-HT2A antagonist

    帕潘立酮, 99%, 高效D25HT2A拮抗劑

    144598-75-4

    10 mg

    50 mg

    144809

    Sumatriptan succinate, 98%, 5-HT1 receptor agonist

    琥珀酸舒馬曲普坦, 98%, 5-HT1 受體激動劑

    103628-48-4

    100 mg

    500 mg

    522188

    Tropisetron monohydrochloride, 99%, 5-HT3 receptor antagonist and α7-nicotinic receptor agonist

    鹽酸托烷司瓊, 99%, 5-HT3受體拮抗劑和α7-煙堿受體激動劑

    105826-92-4

    1 g

    5 g

    186095

    Ziprasidone hydrochloride monohydrate, 99%, a novel and potent dopamine and serotonin (5-HT) receptor antagonist

    齊拉西酮鹽酸鹽一水合物, 99%, 有效的dopamine serotonin (5-HT) receptor的拮抗劑

    138982-67-9

    250 mg

    1 g

                     

                                           Figure1                                                                                      Figure2

    Figure1: Structure of Lamotrigine (185928)[1] 

    Figure2: Interactions of Lamotrigine(185928) with the binding pocket (subdomain IB)[1]

     References

    [1] Poureshghi F, Ghandforoushan P, Safarnejad A, et al. Interaction of an antiepileptic drug, lamotrigine with human serum albumin (HSA): Application of spectroscopic techniques and molecular modeling methods[J]. Journal of Photochemistry and Photobiology B: Biology, 2017, 166: 187-192.

    [2]Yatham L N, Beaulieu S, Schaffer A, et al. Optimal duration of risperidone or olanzapine adjunctive therapy to mood stabilizer following remission of a manic episode: A CANMAT randomized double-blind trial[J]. Molecular psychiatry, 2016, 21(8): 1050-1056.

     

    產品編號

    中英文名稱

    CAS

    包裝規格

    163651

    (+)-Bicuculline, 99.5%, GABAA antagonist

    (+)-荷包牡丹堿, 99.5%, GABAA 拮抗劑

    485-49-4

    25 mg

    100 mg

    240627

    Candesartan cilexetil, 98%, ATR antagonist

    坎地沙坦酯, 98%, ATR 拮抗劑

    145040-37-5

    50 mg

    100 mg

    500 mg

    410760

    Cyproterone acetate, 98%, an androgen receptor (AR) antagonist

    環丙孕酮醋酸鹽, 98%, 一種雄激素受體拮抗劑

    427-51-0

    50 mg

    250 mg

    1 g

    195685

    Leuprorelin acetate, 98%, an agonist at pituitary GnRH receptors

    醋酸亮丙瑞林, 98%, 一種垂體促性腺激素受體抑制劑

    74381-53-6

    5 mg

    25 mg

    408413

    Tropicamide, 99%, potent selective M4 antagonist

    托品酰胺, 99%, 有效選擇性M4拮抗劑

    1508-75-4

    10 g

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